Bioactive small molecules are organic compounds that have a low molecular weight (900 daltons). Most pharmaceutical drugs are small molecules. Larger structures such as nucleic acids, proteins, and many polysaccharides are not small molecules.
Iodoacetamide is a thiol reagent and can inhibit glycolysis and can be used to study the role of cysteine residues in enzymology. Iodoacetamide is an alkylating reagent for cysteine residues in...
Rezafungin Acetate (syn: biafungin acetate) is the acetate salt of Rezafungin, a semi-synthetic, next-generation, broad-spectrum echinocandin. It is antifungal agent with activity against...
Oteseconazole is a novel tetrazole that has activity against bacteria causing vulvovaginal candidiasis (RVVC). It is a selective inhibitor of fungal cytochrome P450 enzyme 51 (CYP51). The tetrazole...
Levamisole Hydrochloride, USP is the pure levorotatory (L) isomer of Tetramisole. This imidazothiazole is responsible for almost all of the antiparasitic activity of this product. It is a nicotinic...
Enmetazobactam is a penicillanic acid sulfone extended-spectrum β-lactamase (ESBL) inhibitor. It is an N-methylated tazobactam derivative ideveloped at Orchid Pharma (India) and then out-licensed to...
Zoliflodacin is a spiropyrimidinetrione antibiotic belonging to the fluoroquinolone class. It is a bacterial DNA gyrase inhibitor with in vitro antibacterial activity against key Gram-positive,...
Gepotidacin is a novel triazaacenaphthylene bacterial type II topoisomerase inhibitor. The compound was developed by GlaxoSmithKline (London, UK) and has broad-spectrum in vitro activity against...
Danofloxacin is a broad-spectrum antibiotic and third-generation fluoroquinolone class. It was developed by Pfizer and is a synthetic analog of ciprofloxacin. It was introduced in 1991 for pathogens...
Cefetamet Sodium is the sodium salt of Cefetamet, a broad-spectrum third-generation cephalosporin antibiotic. It is classified as a 'aminothiazolyl imimomethoxy cephalosporin' since it has both...
Cefetamet is a broad-spectrum, third-generation cephalosporin antibiotic. It is classified as a 'aminothiazolyl imimomethoxy cephalosporin' since it has both methyl and...
Tinidazole is a broad-spectrum second-generation 5-nitroimidazole antibiotic and synthetic antiprotozoal agent introduced in 1969. This imidazole derivative is used against bacteria, protozoa and...
Ornidazole is a nitroimidazole antibiotic and antiparasitic agent, with broad-spectrum antiprotozoan and anti-aerobic activity. It was synthsized by Hoffmann-La-Roche (1966) and was first introduced...
